|
Product |
Laboratory |
Substance |
Dosage |
Contains |
Price |
Order! |
|
Nolvadex 20 |
Astra-Zeneca |
Tamoxifen citrate |
20 mg./tab |
30 tabs |
$39.00 |
 |
Nolvadex®, a trade name for the drug
tamoxifen citrate, is a non-steroidal agent that demonstrates potent
antiestrogenic properties. The drug is technically an estrogen
agonist/antagonist, which competitively binds to estrogen receptors
in various target tissues. With the tamoxifen molecule bound to this
receptor, estrogen is blocked from exerting any action, and an
antiestrogenic effect is achieved. Since many forms of breast cancer
are responsive to estrogen, the ability of tamoxifen citrate to
block its action in such cells has proven to be a very effective
treatment. It is also utilized successfully as a preventative
measure, taken by people with an extremely high familial tendency
for breast cancer. While Nolvadex® is effective against estrogen, it
is not our strongest available remedy. We now have the drug
Arimidex® available to us, which
notably prevents estrogen from being manufactured in the first
place. Altering the effect of estrogen in the female body can cause
a level of discomfort, so antiestrogens are most bearable when used
after the point of menopause. Since Nolvadex® is milder in
comparison, it is more widely applicable and usually the first
treatment option.
As discussed earlier in this book, an enzyme in the male body (aromatase)
is capable of altering testosterone to form estradiol. The structure
of estrogen is actually quite similar to testosterone, so its
presence in the male body is not all that remarkable. Since this
same enzyme can also aromatize many anabolic/androgenic steroids,
the buildup of estrogens can be an important concern during intake.
High levels can cause a number of unwanted side effects, a primary
worry being gynecomastia or the development of female breast tissue
in men. This can be first noticed by the appearance of swelling or a
small lump under the nipple. If left to progress it can turn into a
very unsightly development of tissue, often an irreversible
occurrence without surgery. Estrogen can also lead to an increase in
the level of water retained in the body. The result here can be a
notable loss of definition, the muscles beginning to look smooth and
bloated due to the retention of subcutaneous fluid. Fat storage may
also be increased as estrogen levels rise. This hormone is in fact
the primary reason women have a higher body fat percentage, and
different fat distribution (hips/thighs) than men. Individuals
sensitive to the effects of estrogen will usually be sure to have an
antiestrogen on hand when taking problematic steroids, so as to
minimize the impact of related side effects. It is also of note that
when estrogen and body fat levels are normal, administering Nolvadex®
(both Men and Women) can increase the look of hardness and
definition the muscles.
|
Product |
Laboratory |
Substance |
Dosage |
Contains |
Price |
Order! |
|
Nolvadex 20 |
Astra-Zeneca |
Tamoxifen citrate |
20 mg./tab |
30 tabs |
$39.00 |
 |
|